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ICONC13707 GDC-0941 bismesylate (957054-30-7)
 
 
Catalog No.: C13707
CAS No.: 957054-30-7
Synonym: Pictilisib; GDC 0941; GDC0941
Chemical Name:

2-(1H-Indazol-4-yl)-6-(4-methanesulfonyl-piperazin-1ylmethyl)-4-morpholin-4-yl-thieno[3,2-d]pyrimidine bismesylate
Molecular Formula:

C23H27N7O3S2.2CH3SO3H
Molecular Weight: 705.83
 
Technical Data:
Appearance: White solid
Solubility: Soluble in DMSO
Purity: >99%
Storage: at +4℃
Original QC Data:
Shipping Conditions: Ambient Temp.
 
Price and Availability of GDC-0941 bismesylate:

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Price

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10mg 

USD

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50mg 

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In stock 

100mg 

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Contact us for competitive discounts on bulk quantities
 
Biological Activity:

A potent, selective, orally bioavailable inhibitor of PI3K  and being evaluated in human clinical trials for the treatment of cancer.
 
References:
Wallin JJ  et al. GDC-0941, a novel class I selective PI3K inhibitor, enhances the efficacy of docetaxel in human breast cancer models by increasing cell death in vitro and in vivo. Clin Cancer Res 18:3901-11 (2012).
 
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